Biochemical Pharmacology of the Sigma|1 Receptor

Biochemical Pharmacology of the Sigma-1 Receptor - PubMed

The sigma-1 receptor (S1R) is a 223 amino acid two transmembrane (TM) pass protein. It is a non-ATP-binding nonglycosylated ligand-regulated molecular ...

Biochemical Pharmacology of the Sigma-1 Receptor

In vivo, the sigma-1 receptor is proposed to bind agonists as a dimer and/or monomer (or the agonists create functionally active dimers and/or ...

Biochemical Pharmacology of the Sigma-1 Receptor

The sigma-1 receptor (S1R) is a 223 amino acid two transmem- brane (TM) pass protein. It is a non-ATP-binding nonglycosylated ligand-regulated molecular ...

The pharmacology of sigma-1 receptors - PubMed

... sigma-1 receptor at the endoplasmic reticulum might relate to so many diseases. We found that the most prominent action of sigma-1 receptors in biological ...

Biochemical Pharmacology of the Sigma-1 Receptor - ResearchGate

The Sigma-1 Receptor (S1R) is a small, ligand-regulated integral membrane protein involved in cell homeostasis and the cellular stress response.

Table 2 from Biochemical Pharmacology of the Sigma-1 Receptor

Table 2: Amino acid residues of the sigma-1 receptor affected by mutation - "Biochemical Pharmacology of the Sigma-1 Receptor"

Molecular cloning and pharmacological characterization of the rat ...

1 August 2001, Pages 349-355. Biochemical Pharmacology. Molecular cloning and pharmacological characterization of the rat sigma1 receptor. Author links open ...

Biochemical Pharmacology | Journal | ScienceDirect.com by Elsevier

Quantities used for concentration- and dose-response experiments should vary logarithmically, e.g., 1 ... The 6th International Ah Receptor Meeting: Research, ...

Comparative biochemical pharmacology of central nervous system ...

(1986) The D-1 dopamine receptor antagonist SCH 23390 also interacts potently with brain serotonin (5-HT2) receptors.Eur. J. Pharmacol. 129, 367–370. Article ...

Sigma receptors | Other protein targets

(2016) Biochemical Pharmacology of the Sigma-1 Receptor. Mol Pharmacol, 89 (1): 142-53. [PMID:26560551]. de Medina P, Paillasse MR, Ségala G, Khallouki F ...

Biochemical pharmacology of the vanilloid receptor TRPV1 - 2004

The vanilloid (capsaicin) receptor; transient receptor potential channel, vanilloid subfamily member 1 (TRPV1), is subjected to multiple interacting levels of ...

Biochemical Pharmacology Core | Lewis Katz School of Medicine

Radioligand binding to mu, delta and kappa opioid receptors (MOPR, DOPR, KOPR), the nociceptin / orphanin FQ receptor (NOPR), as well as to the dopamine, sigma, ...

Biochemical pharmacology of serotonin receptor subtypes

This article discusses the pharmacological basis for applying advances in serotonin receptor subtyping to the development of novel psychiatric ...

Receptor (biochemistry) - Wikipedia

In biochemistry and pharmacology, receptors are chemical structures ... These signals are typically chemical messengers which bind to a receptor ...

The biochemical pharmacology of metabotropic glutamate receptors

Biochem Soc Trans (1993) 21 (1): 97–102. https://doi.org/10.1042/bst0210097. Article history.

Development of a Novel σ1 Receptor Biosensor Based on Its ...

Biochemical pharmacology of the sigma-1 receptor. Chu, Uyen B.; Ruoho, Arnold E. Molecular Pharmacology (2016), 89 (1), 142-153CODEN: MOPMA3 ...

Functionally selective cannabinoid receptor signalling

revealing that biological activities modulated by cannabinoid. Biochemical Pharmacology 80 (2010) 1–12. A R T I C L E I N F O. Article history: Received 4 ...

Biochemical Pharmacology of Dopamine Receptors - SpringerLink

Memo, M., Lovenberg, W., and Hanbauer, 1., Agonist-induced sub-sensitivity of adenylate cyclase coupled with a dopamine receptor in slices from rat corpus ...

Molecular and biochemical pharmacology of the histamine H4 ...

Bell JK, McQueen DS, Rees JL (2004). Involvement of histamine H4 and H1 receptors in scratching induced by histamine receptor agonists in Balb C ...

Neuronal Sigma-1 Receptors: Signaling Functions and Protective ...

... receptor: biochemical and physiological evidences, consequences ... Pharmacological profiling of sigma 1 receptor ligands by novel receptor homomer assays.